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Day One Biopharmaceuticals, Inc.

Pipeline3 assets

  • TovorafenibDAY101 / OJEMDA / RAF / MAPK pathway / Oral small-molecule type II RAF inhibitor / Oncology
    BRAF-altered relapsed pLGGApprovedOJEMDA received FDA accelerated approval; FIREFLY-1 pivotal Phase 2 follow-up ongoing/disclosedU.S.Frontline RAF-altered pLGGPhase 3 / RegistrationalFIREFLY-2 pivotal Phase 3
  • Emiltatug ledadotinEmi-Le / B7-H4 / Antibody-drug conjugate (ADC) / Oncology
    Adenoid cystic carcinoma (ACC), adult and pediatric solid tumorsPhase 1B7-H4-targeted ADC; Phase 1 data anticipated mid-2026 per company investor materials
  • DAY301MTX-13 / CB-002 / PTK7 / Antibody-drug conjugate (ADC) / Oncology
    Adult and pediatric solid tumorsPhase 1Phase 1a data anticipated 2H 2026 per company investor materials

Latest news6 items

All news

Day One Completes Acquisition of Mersana Therapeutics

Acquisition expands Day One’s pipeline with clinical-stage antibody drug conjugate (ADC) emiltatug ledadotin (Emi-Le) targeting rare cancer adenoid cystic carcinoma (ACC) BRISBANE, Calif., Jan. 06, 2026 (GLOBE NEWSWIRE) -- Day One Biopharmaceuticals, Inc.

Day One to Present at the 44th Annual J.P. Morgan Healthcare Conference

BRISBANE, Calif., Dec. 16, 2025 (GLOBE NEWSWIRE) -- Day One Biopharmaceuticals, Inc. (Nasdaq: DAWN) (“Day One” or the “Company”), a biopharmaceutical company dedicated to developing and commercializing targeted therapies for people of all ages with life-threatening diseases, today announced that

Day One Biopharmaceuticals, Inc. • Endpoint Arena